broad_id
string
depmap_id
string
ccle_name
string
screen_id
string
upper_limit
int64
lower_limit
float64
slope
float64
r2
float64
auc
float64
ec50
float64
ic50
float64
name
string
moa
string
target
string
disease.area
string
indication
string
smiles
string
phase
string
passed_str_profiling
bool
row_name
string
BRD-K71847383-001-12-5
ACH-000288
BT549_BREAST
HTS002
1
1.810211
0.111243
-0.003031
1.302289
9.260129
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000288
BRD-K71847383-001-12-5
ACH-000415
BICR6_UPPER_AERODIGESTIVE_TRACT
HTS002
1
1.409581
0.120752
-0.061802
1.169222
1.550463
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000415
BRD-K71847383-001-12-5
ACH-000228
BICR31_UPPER_AERODIGESTIVE_TRACT
HTS002
1
1.982005
-0.164109
0.131114
1.369119
0.003036
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000228
BRD-K71847383-001-12-5
ACH-000977
LNCAPCLONEFGC_PROSTATE
HTS002
1
1.176368
5.44413
-0.142784
1.088256
0.077814
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000977
BRD-K71847383-001-12-5
ACH-000397
TEN_ENDOMETRIUM
HTS002
1
2.26404
-0.082945
0.010249
1.492828
0.000329
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000397
BRD-K71847383-001-12-5
ACH-000565
RCM1_LARGE_INTESTINE
HTS002
1
1.590267
0.109949
-0.042492
1.302732
0.048366
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000565
BRD-K71847383-001-12-5
ACH-000209
SNU1079_BILIARY_TRACT
HTS002
1
1.555816
0.12506
-0.095405
1.29347
0.031018
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000209
BRD-K71847383-001-12-5
ACH-000927
BT474_BREAST
HTS002
1
1.595816
0.117463
0.035402
1.243364
1.988602
null
cytarabine
ribonucleotide reductase inhibitor
POLA1, POLB, POLD1, POLE
hematologic malignancy
acute lymphoblastic leukemia (ALL), chronic lymphocytic leukemia (CLL), acute myeloid leukemia (AML), non-Hodgkin lymphoma (NHL)
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1, Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1
Launched
true
ACH-000927
BRD-A98990573-003-01-3
ACH-000879
MFE296_ENDOMETRIUM
HTS002
1
2.406651
-0.073609
-0.123828
1.718502
0.141302
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000879
BRD-A98990573-003-01-3
ACH-000320
PSN1_PANCREAS
HTS002
1
2.153169
0.01822
-0.015702
1.565786
0.611409
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000320
BRD-A98990573-003-01-3
ACH-001145
OC316_OVARY
HTS002
1
1.930698
-0.128307
0.013193
1.525007
0.621301
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-001145
BRD-A98990573-003-01-3
ACH-000873
KYSE270_OESOPHAGUS
HTS002
1
1.663819
0.09446
0.017444
1.333858
0.068841
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000873
BRD-A98990573-003-01-3
ACH-000855
KYSE150_OESOPHAGUS
HTS002
1
2.443731
0.035814
-0.07384
1.461459
119,125,404.206814
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000855
BRD-A98990573-003-01-3
ACH-000913
ESS1_ENDOMETRIUM
HTS002
1
1.986984
0.276565
0.206415
1.455895
0.147025
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000913
BRD-A98990573-003-01-3
ACH-000558
A172_CENTRAL_NERVOUS_SYSTEM
HTS002
1
2.393393
-0.198751
-0.162024
1.581816
0.012899
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000558
BRD-A98990573-003-01-3
ACH-000593
BC3C_URINARY_TRACT
HTS002
1
2.131649
0.0142
0.017346
1.544465
15.994651
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000593
BRD-A98990573-003-01-3
ACH-000488
TE11_OESOPHAGUS
HTS002
1
1.403471
-0.146593
0.056054
1.249404
2.389566
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000488
BRD-A98990573-003-01-3
ACH-000832
CAL27_UPPER_AERODIGESTIVE_TRACT
HTS002
1
1.806094
-0.136659
-0.006901
1.462856
0.753831
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000832
BRD-A98990573-003-01-3
ACH-000781
NCIH2023_LUNG
HTS002
1
2.116241
0.013514
-0.043877
1.562774
0.022735
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000781
BRD-A98990573-003-01-3
ACH-000833
RH30_SOFT_TISSUE
HTS002
1
1.704559
-0.009088
-0.044286
1.355226
0.492545
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000833
BRD-A98990573-003-01-3
ACH-000137
8MGBA_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.912906
0.080341
-0.114723
1.510014
0.004002
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000137
BRD-A98990573-003-01-3
ACH-000632
HS944T_SKIN
HTS002
1
1.808378
-0.002097
-0.205969
1.405029
0.567232
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000632
BRD-A98990573-003-01-3
ACH-000630
YD8_UPPER_AERODIGESTIVE_TRACT
HTS002
1
1.659657
0.212536
-0.070869
1.347965
0.044491
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000630
BRD-A98990573-003-01-3
ACH-000266
SNU213_PANCREAS
HTS002
1
2.197751
-0.07709
-0.101426
1.680144
2.812235
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000266
BRD-A98990573-003-01-3
ACH-000047
GCIY_STOMACH
HTS002
1
1.169463
-0.063424
-0.122913
1.0977
10.520899
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000047
BRD-A98990573-003-01-3
ACH-000273
SF539_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.781141
-0.17458
-0.010169
1.428111
0.251615
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000273
BRD-A98990573-003-01-3
ACH-000682
SNU1066_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.906513
0.253387
-0.001659
0.940251
0.006255
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000682
BRD-A98990573-003-01-3
ACH-000359
MG63_BONE
HTS002
1
0.678547
0.290458
-0.106625
0.753177
0.000707
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000359
BRD-A98990573-003-01-3
ACH-000846
FADU_UPPER_AERODIGESTIVE_TRACT
HTS002
1
0.687044
0.113647
0.01733
0.945489
92,317.295283
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000846
BRD-A98990573-003-01-3
ACH-000804
NB1_AUTONOMIC_GANGLIA
HTS002
1
1.03215
-0.193507
-0.043366
1.018095
0.31676
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000804
BRD-A98990573-003-01-3
ACH-000609
SF126_CENTRAL_NERVOUS_SYSTEM
HTS002
1
0.722635
-0.381214
-0.036432
0.8183
0.651099
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000609
BRD-A98990573-003-01-3
ACH-000974
SNGM_ENDOMETRIUM
HTS002
1
1.995466
-0.168702
-0.009664
1.500396
0.083533
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000974
BRD-A98990573-003-01-3
ACH-000987
MEWO_SKIN
HTS002
1
1.650375
0.375233
0.301196
1.303564
0.122256
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000987
BRD-A98990573-003-01-3
ACH-000787
LXF289_LUNG
HTS002
1
1.532402
0.858926
0.228983
1.255558
0.095433
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000787
BRD-A98990573-003-01-3
ACH-000561
TT_OESOPHAGUS
HTS002
1
1.274219
-0.017798
0.004438
1.158504
3,764,418.111465
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000561
BRD-A98990573-003-01-3
ACH-000212
CAL120_BREAST
HTS002
1
1.842452
0.128951
0.033742
1.405999
0.139407
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000212
BRD-A98990573-003-01-3
ACH-000753
JMSU1_URINARY_TRACT
HTS002
1
1.49449
-0.236912
0.022282
1.270752
0.190536
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000753
BRD-A98990573-003-01-3
ACH-000305
ECGI10_OESOPHAGUS
HTS002
1
1.61547
-0.052329
-0.029299
1.358002
43.970646
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000305
BRD-A98990573-003-01-3
ACH-000138
CFPAC1_PANCREAS
HTS002
1
1.753365
0.257979
0.130517
1.380023
0.072298
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000138
BRD-A98990573-003-01-3
ACH-000250
KMRC20_KIDNEY
HTS002
1
1.494624
0.395246
0.190654
1.209002
0.215924
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000250
BRD-A98990573-003-01-3
ACH-000856
CAL51_BREAST
HTS002
1
1.735025
-0.228678
0.10814
1.285053
0.008714
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000856
BRD-A98990573-003-01-3
ACH-000046
ACHN_KIDNEY
HTS002
1
2.014146
0.0271
-0.020242
1.465787
32.507875
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000046
BRD-A98990573-003-01-3
ACH-000878
HCC15_LUNG
HTS002
1
1.964366
0.135892
0.020902
1.235052
425.682928
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000878
BRD-A98990573-003-01-3
ACH-000766
NCIH1648_LUNG
HTS002
1
1.552756
0.044905
0.023289
1.263833
0.595469
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000766
BRD-A98990573-003-01-3
ACH-000014
HS294T_SKIN
HTS002
1
1.866487
-0.441467
0.082457
1.491065
0.177963
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000014
BRD-A98990573-003-01-3
ACH-000701
RMUGS_OVARY
HTS002
1
1.93928
-0.108778
0.062088
1.4956
0.221216
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000701
BRD-A98990573-003-01-3
ACH-000884
MDAMB435S_SKIN
HTS002
1
1.561581
-0.062436
-0.00177
1.511362
1,325,035,067,871,792
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000884
BRD-A98990573-003-01-3
ACH-000037
S117_SOFT_TISSUE
HTS002
1
2.610757
-0.322145
0.057094
1.353067
0.000771
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000037
BRD-A98990573-003-01-3
ACH-000502
TCCPAN2_PANCREAS
HTS002
1
1.791147
0.046662
-0.052582
1.445164
0.000344
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000502
BRD-A98990573-003-01-3
ACH-000886
NCIH2009_LUNG
HTS002
1
1.824982
-0.040267
0.016273
1.40362
0.02675
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000886
BRD-A98990573-003-01-3
ACH-000035
NCIH1650_LUNG
HTS002
1
1.275007
0.014939
-0.127125
1.13901
0.017995
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000035
BRD-A98990573-003-01-3
ACH-000661
WM1799_SKIN
HTS002
1
1.373218
0.176351
0.033827
1.191805
0.055892
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000661
BRD-A98990573-003-01-3
ACH-000391
MHHES1_BONE
HTS002
1
1.321053
-0.094279
-0.007156
1.150176
0.019392
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000391
BRD-A98990573-003-01-3
ACH-000843
HARA_LUNG
HTS002
1
1.976587
-0.10598
0.080794
1.457676
0.023278
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000843
BRD-A98990573-003-01-3
ACH-000711
JIMT1_BREAST
HTS002
1
1.948984
0.184036
0.071032
1.52785
0.021135
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000711
BRD-A98990573-003-01-3
ACH-000232
U251MG_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.542617
0.219233
0.156442
1.261488
0.112082
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000232
BRD-A98990573-003-01-3
ACH-000060
PANC1005_PANCREAS
HTS002
1
1.801116
0.105156
-0.010876
1.297048
13.271048
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000060
BRD-A98990573-003-01-3
ACH-000322
HT144_SKIN
HTS002
1
2.744352
0.163127
0.199069
1.879861
0.069734
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000322
BRD-A98990573-003-01-3
ACH-000736
SNU601_STOMACH
HTS002
1
1.354943
-0.272767
-0.153729
1.097497
0.001394
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000736
BRD-A98990573-003-01-3
ACH-000809
KYSE410_OESOPHAGUS
HTS002
1
1.745682
0.225432
0.22769
1.36529
0.09516
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000809
BRD-A98990573-003-01-3
ACH-000747
NCIH1703_LUNG
HTS002
1
1.930434
8.051284
0.358434
1.331938
0.313671
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000747
BRD-A98990573-003-01-3
ACH-000364
U2OS_BONE
HTS002
1
1.623598
-0.010964
-0.091907
1.340628
1,739,143.771505
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000364
BRD-A98990573-003-01-3
ACH-000679
OE19_OESOPHAGUS
HTS002
1
1.981374
0.064406
-0.099249
1.496815
0.052841
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000679
BRD-A98990573-003-01-3
ACH-000985
LS411N_LARGE_INTESTINE
HTS002
1
0.880762
1.193111
-0.100253
0.951954
0.2018
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000985
BRD-A98990573-003-01-3
ACH-000441
SH4_SKIN
HTS002
1
1.660765
-1.079061
0.253114
1.40478
0.236411
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000441
BRD-A98990573-003-01-3
ACH-001113
LC1SQSF_LUNG
HTS002
1
1.671028
-0.623007
0.292925
1.414209
0.277152
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-001113
BRD-A98990573-003-01-3
ACH-000620
JHH1_LIVER
HTS002
1
6.052251
-1.201168
0.02801
1.085837
0.000172
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000620
BRD-A98990573-003-01-3
ACH-000853
NCIH661_LUNG
HTS002
1
1.797602
0.127079
0.052302
1.374245
0.212531
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000853
BRD-A98990573-003-01-3
ACH-000102
GMS10_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.341286
0.008135
-0.015857
1.171228
0.033644
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000102
BRD-A98990573-003-01-3
ACH-000648
NCIH28_PLEURA
HTS002
1
2.670765
0.188381
0.080214
1.576709
2.930078
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000648
BRD-A98990573-003-01-3
ACH-001321
TT_THYROID
HTS002
1
1.600621
0.319511
0.229367
1.325862
0.04134
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-001321
BRD-A98990573-003-01-3
ACH-000279
EWS502_BONE
HTS002
1
1.392272
-0.116253
-0.144175
1.318358
29,553.560728
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000279
BRD-A98990573-003-01-3
ACH-000172
TM87_SOFT_TISSUE
HTS002
1
1.191382
0.018894
-0.123475
1.095645
0.082241
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000172
BRD-A98990573-003-01-3
ACH-001128
MON_SOFT_TISSUE
HTS002
1
2.837286
1.31773
0.351164
2.530067
0.002812
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-001128
BRD-A98990573-003-01-3
ACH-000437
SW1088_CENTRAL_NERVOUS_SYSTEM
HTS002
1
2.464921
-0.161799
0.021702
1.483223
0.00079
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000437
BRD-A98990573-003-01-3
ACH-000207
DETROIT562_UPPER_AERODIGESTIVE_TRACT
HTS002
1
2.28056
-0.229442
0.28321
1.603477
0.044971
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000207
BRD-A98990573-003-01-3
ACH-000260
SKNAS_AUTONOMIC_GANGLIA
HTS002
1
1.546904
-0.151411
-0.033138
1.293755
0.218017
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000260
BRD-A98990573-003-01-3
ACH-000019
MCF7_BREAST
HTS002
1
1.46547
-0.100758
-0.017226
1.302785
41.859975
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000019
BRD-A98990573-003-01-3
ACH-000582
COLO741_SKIN
HTS002
1
1.448067
-0.27547
-0.096245
1.379457
79.715214
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000582
BRD-A98990573-003-01-3
ACH-000990
HEC108_ENDOMETRIUM
HTS002
1
1.570831
-0.088779
-0.037785
1.476341
8,069,214.118125
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000990
BRD-A98990573-003-01-3
ACH-000592
TM31_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.369895
0.257976
-0.091276
1.250242
0.003161
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000592
BRD-A98990573-003-01-3
ACH-000368
SNU1105_CENTRAL_NERVOUS_SYSTEM
HTS002
1
1.494473
-0.146671
-0.066263
1.342403
24.62497
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000368
BRD-A98990573-003-01-3
ACH-000517
SNU410_PANCREAS
HTS002
1
2.405004
-0.306842
-0.271216
1.315484
0.00073
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000517
BRD-A98990573-003-01-3
ACH-000374
HCC1143_BREAST
HTS002
1
1.971707
-0.160977
0.131079
1.41006
0.010041
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000374
BRD-A98990573-003-01-3
ACH-000527
OVISE_OVARY
HTS002
1
1.663536
0.24615
-0.080177
1.479834
0.001039
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000527
BRD-A98990573-003-01-3
ACH-000091
OV56_OVARY
HTS002
1
1.298686
-0.17482
-0.14306
1.177357
0.778295
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000091
BRD-A98990573-003-01-3
ACH-000759
MDAMB175VII_BREAST
HTS002
1
1.010161
-0.128943
-0.129627
1.006279
3.668881
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000759
BRD-A98990573-003-01-3
ACH-000417
PANC0813_PANCREAS
HTS002
1
1.813245
0.270191
-0.044787
1.365034
0.185574
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000417
BRD-A98990573-003-01-3
ACH-000308
EFO21_OVARY
HTS002
1
1.413574
0.086931
-0.024889
1.224231
0.01085
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000308
BRD-A98990573-003-01-3
ACH-000991
SNU81_LARGE_INTESTINE
HTS002
1
1.966944
0.040441
-0.016903
1.22707
411,647,219,914.019
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000991
BRD-A98990573-003-01-3
ACH-000948
2313287_STOMACH
HTS002
1
1.177057
-0.502442
-0.090841
1.118802
0.594219
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000948
BRD-A98990573-003-01-3
ACH-000481
NCIH2170_LUNG
HTS002
1
1.87338
0.008744
-0.017357
1.443936
0.001754
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000481
BRD-A98990573-003-01-3
ACH-000771
BICR56_UPPER_AERODIGESTIVE_TRACT
HTS002
1
1.819329
-0.09418
0.07333
1.393692
0.033634
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000771
BRD-A98990573-003-01-3
ACH-000159
OSRC2_KIDNEY
HTS002
1
1.262509
0.147054
0.025325
1.116855
0.372107
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000159
BRD-A98990573-003-01-3
ACH-000929
NCIH2110_LUNG
HTS002
1
3.663559
0.881271
0.148348
1.129812
21.129337
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000929
BRD-A98990573-003-01-3
ACH-000118
HUPT3_PANCREAS
HTS002
1
1.794215
-0.358423
0.007789
1.397125
0.078149
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000118
BRD-A98990573-003-01-3
ACH-000482
RERFLCKJ_LUNG
HTS002
1
1.526195
-0.088525
-0.094492
1.184886
0.000069
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000482
BRD-A98990573-003-01-3
ACH-000352
HCC1428_BREAST
HTS002
1
1.507227
0.098268
-0.075063
1.313161
0.000548
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000352
BRD-A98990573-003-01-3
ACH-000235
PANC0403_PANCREAS
HTS002
1
1.894912
-0.030993
-0.148693
1.436389
0.015782
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000235
BRD-A98990573-003-01-3
ACH-000479
KNS81_CENTRAL_NERVOUS_SYSTEM
HTS002
1
2.48851
0.050826
-0.027301
1.494476
77,323.177171
null
epinastine
histamine receptor antagonist
ADRA1A, ADRA2A, HRH1, HRH2, HTR2A, HTR7
ophthalmology
conjunctivitis
NC1=NCC2N1c1ccccc1Cc1ccccc21
Launched
true
ACH-000479